Drug Interactions

Semaglutide Drug Interactions

Also known as: Ozempic, Rybelsus, Wegovy

Semaglutide (Ozempic, Wegovy, Rybelsus) is a GLP-1 receptor agonist approved for type 2 diabetes, weight management, and cardiovascular risk reduction. See the full semaglutide monograph for complete prescribing information.Semaglutide has 1 documented drug interaction in our database, including 0 contraindicated, 0 major, 1 moderate, and 0 minor interactions.

0

Contraindicated

0

Major

1

Moderate

0

Minor

Metformin Hydrochloride(Metformin Hydrochloride)
Moderate

Combining metformin and oral semaglutide can lead to an increased risk of hypoglycemia (low blood sugar) due to their additive glucose-lowering effects. Patients may experience symptoms such as dizziness, sweating, confusion, or tremor. While generally beneficial for blood sugar control, close monitoring is essential.

Mechanism

Both metformin and semaglutide work to lower blood glucose through different mechanisms. Metformin decreases hepatic glucose production and improves insulin sensitivity, while semaglutide, a GLP-1 receptor agonist, stimulates insulin secretion, suppresses glucagon secretion, and slows gastric emptying. Their combined actions can lead to a synergistic reduction in blood glucose levels.

Clinical Management

Monitor blood glucose levels more frequently, especially when initiating or titrating either medication. If hypoglycemia occurs, a dose reduction of one or both medications, particularly any concomitant insulin secretagogues (e.g., sulfonylureas) or insulin, may be necessary. Educate patients on recognizing and treating hypoglycemia.

Evidence: established
Onset: delayed
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For complete prescribing information:

View full Semaglutide monograph →

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